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NEW PHARMACEUTICAL COMPOUNDS

申请公布号:KR20050114603(A)

申请号:KR20057009983

申请日期:2005.06.02

申请公布日期:2005.12.06

申请人:
ORION CORPORATION

发明人:JARVINEN TOMI;NIEMI RIKU;HUUSKONEN JUHANI

分类号:A61P3/06;A61P3/10;C07D233/54;C07D233/56;C07D233/64;(IPC1-7):C07D233/64

主分类号:A61P3/06

摘要:The present invention relates to novel prodrugs of MPV-2426, to methods for preparing said prodrug forms, to pharmaceutical compositions containing such prodrug forms, and to methods for using the prodrug forms. A compound of general formula (I), or pharmaceutically acceptable salts or hydrates thereof, wherein R represents unsubstituted or substituted lower alkyl, unsubstituted or substituted aryl, unsubstituted or substituted cycloalkyl, unsubstituted or substituted heteroaryl, unsubstituted or substituted lower alkylamino or asaturated five or six membered heterocyclic group containing Olle or two nitrogen atoms.

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