IMIDAZO(4,5-B) PYRIDIN-2-YL AMIDES AS KV7 CHANNEL ACTIVATORS
申请公布号:US2016031875(A1)
申请号:US201414776271
申请日期:2014.03.17
申请公布日期:2016.02.04
发明人:Resnick Lynn;Topalov George T.;Boyd Steven A.;Belardi Justin K.;Flentge Charles A.;Hale James S.;Harried Scott S.;Mareska David A.;Zhang Kai;Heap Charles R.;Hadden Mark;Cui Wenge;Decornez Hélène;Liu Shuang
分类号:C07D471/04;C07D519/00
主分类号:C07D471/04
地址:Pittsburgh PA US
摘要:Compounds represented by formula 1 can be potent and/or partially selective for the Kv7.2/7.3 heteromultimer. They may be useful in treating disorders related to seizures, pain, neurotransmitter release, etc.
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