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ORAL COMPOSITION COMPRISING 3-[5-[4-(CYCLOPENTYLOXY) -2-HYDROXYBENZOYL]-2-[(3-HYDROXY-1,2-BENZISOXAZOL-6- YL)METHOXY]PHENYL]PROPIONIC ACID OR SALT THEREOF.

申请公布号:MX2008015015(A)

申请号:MX20080015015

申请日期:2007.05.25

申请公布日期:2008.12.05

申请人:
TOYAMA CHEMICAL CO., LTD.

发明人:SAHOE KAKUDA;TATSUHITO YAHATA;MASASHI KANEKO

分类号:A61K31/423;A61K9/08;A61K9/20;A61K9/48;A61K47/02;A61K47/18;A61K47/32;A61P29/00

主分类号:A61K31/423

摘要:<p>An oral composition comprising 3-[5-[4- (cyclopentyloxy)-2-hydroxybenzoyl]-2-[(3-hydroxy-1,2- benzisoxazol-6-yl)methoxy]phenyl]propionic acid or a salt thereof and polyvinylpyrrolidone. The oral composition is useful as a pharmaceutical composition for oral application having the following properties (1) to (3): (1) no new-type facility is required for the production of the composition; (2) the composition can be produced by a simple process; and (3) the composition can be dissolved stably in the gastrointestinal tract even when the pH value in the gastrointestinal tract varies and therefore is improved in gastrointestinal adsorption.</p>

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