NOVEL LAPACHONE COMPOUNDS AND METHODS OF USE THEREOF
申请公布号:EP1567515(A2)
申请号:EP20030786941
申请日期:2003.11.18
申请公布日期:2005.08.31
发明人:JIANG, ZHIWEI;REDDY, DASHARATHA;ACKERMAN, SAMUEL, K.;SALVESEN, JUNE;SUN, XIANGAO;LI, YOUZHI;LI, CHIANG
分类号:C07D327/06;A61K;A61K31/38;A61K31/382;A61K31/385;A61P35/00;C07D307/92;C07D311/92;C07D333/74;C07D335/08;C07D335/10
主分类号:C07D327/06
摘要:The invention provides lapachone analogs and derivatives as well as methods of use thereof. These compounds can be used in pharmaceutical compositions for the treatment or prevention of cell proliferation disorders. These compounds can also be used in the treatment or prevention of psoriasis or cancer or precancerous conditions.