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PROCESS FOR PREPARING SPARINGLY WATER-SOLUBLE SALTS OF PENICILLANIC ACID 1,1-DIOXIDE

申请公布号:KR850001353(B1)

申请号:KR19820000413

申请日期:1982.02.01

申请公布日期:1985.09.21

申请人:
PFIZER INC.

发明人:ARMSTRONG WILLIAM WELLESLEY;MOPPETT CHARLES EDWARD;WINDISCH WENDELL WILLIAM

分类号:C07D499/897;A61K31/43;A61P31/04;C07D499/00;C07D499/14;C07D499/24;C07D499/86;C07D499/87;C07D499/893;(IPC1-7):C07D499/14

主分类号:C07D499/897

摘要:N,N-dibenzyl ethylenediamine, N-benzyl-2-phenylethylamine, and dibenzylamine were prepd. The salts are sparingly soluble in water, and are of value as slow-release forms of penicillanic acid 1,1-dioxide, in conjunction with sparingly soluble -lactam antibiotics in chemotherapy of bacterial infections in mammals.

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