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包括亚甲基蓝(MTC)之二氨基吩噻嗪鎓化合物的化学合成方法;METHODS OF CHEMICAL SYNTHESIS OF DIAMINOPHENOTHIAZINIUM COMPOUNDS INCLUDING METHYLTHIONINIUM CHLORIDE (MTC)

申请公布号:TW201520202

申请号:TW103134782

申请日期:2014.10.06

申请公布日期:2015.06.01

申请人:
威斯塔实验室公司 WISTA LABORATORIES LTD.

发明人:辛克莱儿詹姆士彼得 SINCLAIR, JAMES PETER;尼可莎拉露意斯 INCOLL, SARAH LOUISE;史托瑞约翰马份大衞 STOREY, JOHN MERVYN DAVID

分类号:C07D279/18(2006.01);C07D279/34(2006.01);A61K31/5415(2006.01)

主分类号:C07D279/18(2006.01)

代理人:蔡坤财李世章

地址:新加坡 SG

摘要:本发明提供合成及纯化包括亚甲基蓝(MTC)(亦称为亚甲蓝)的某些3,7-二氨基-吩噻嗪-5-鎓化合物(在本文中称为「二氨基吩噻嗪鎓化合物」)之方法。;Methods of synthesizing and purifying certain 3,7-diamino-phenothiazin-5-ium compounds (referred to herein as “diaminophenothiazinium compounds”) including Methythioninium Chloride (MTC) (also known as Methylene Blue) are provided.

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