一种微管蛋白聚合剂多肽及其应用
申请公布号:CN103288926A
申请号:CN201310208866.7
申请日期:2013.05.30
申请公布日期:2013.09.11
发明人:罗瑞雪
分类号:C07K7/08(2006.01)I;A61K38/10(2006.01)I;A61P35/02(2006.01)I
主分类号:C07K7/08(2006.01)I
地址:215000 江苏省苏州市高新区竹园路209号
摘要:本发明涉及药物领域,具体涉及具有促进微管蛋白聚合,治疗治疗急性淋巴细胞性白血病的多肽。其序列为EVVPFQEVWGRSYCRA是全新的序列,它们可以在1微摩尔水平上体外促进微管蛋白聚合,并在体内试验中提高荷瘤小鼠生存率,具有潜在的新药开发价值。
主权项:微管蛋白聚合剂多肽8,其特征在于其序列为EVVPFQEVWGRSYCRA。
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