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PHARMACEUTICAL PREPARATION COMPRISING BREXPIPRAZOLE AND SUBSTITUTED BETA - CYCLODEXTRIN

申请公布号:WO2013100204(A1)

申请号:WO2012JP84313

申请日期:2012.12.28

申请公布日期:2013.07.04

申请人:
OTSUKA PHARMACEUTICAL CO., LTD.

发明人:HASEGAWA, TETSUYA;TOYOBUKU, HIDEKAZU

分类号:A61K47/48;A61K31/496

主分类号:A61K47/48

摘要:Provided is an aqueous pharmaceutical preparation comprising 7-[4-(4-benzo[b]thiophen-4-yl-piperazin-1-yl)butoxy]-1H-quinolin-2-one (compound (I)) or a salt thereof, which shows improved water solubility of compound (I) or a salt thereof achieved by addition of substituted beta -cyclodextrin. The present invention provides a pharmaceutical preparation comprising compound (I) or a salt thereof, and substituted beta-cyclodextrin.

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