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POLYCYCLIC BETA LACTAM DERIVATIVES FOR THE TREATMENT OF CANCER

申请公布号:WO2012103456(A2)

申请号:WO2012US22935

申请日期:2012.01.27

申请公布日期:2012.08.02

申请人:
BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM;BECKER, FREDERICK, F.;BANIK, BIMAL, K.

发明人:BECKER, FREDERICK, F.;BANIK, BIMAL, K.

分类号:C07D401/04;A61K31/397;A61K31/4523;A61P35/00;C07D205/08

主分类号:C07D401/04

摘要:Provided herein are polycyclic ß-lactam compounds, compositions thereof and methods for the treatment and prevention of diseases such as cancer, including pancreatic cancer and pancreatic cancers resistant to mainline chemotherapeutic agents.

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