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ACTIVATOR FOR PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR .DELTA.

申请公布号:CA2463569(C)

申请号:CA20022463569

申请日期:2002.10.09

申请公布日期:2012.05.15

申请人:
NIPPON CHEMIPHAR CO., LTD.

发明人:SAKUMA, SHOGO;YAMAKAWA, TOMIO;KANDA, TAKASHI;MASUI, SEIICHIRO

分类号:C07D413/06;A61K31/00;A61K31/423;A61K31/427;A61K31/454;A61P3/04;A61P3/06;A61P3/10;A61P9/00;A61P9/10;A61P19/10;A61P25/28;A61P29/00;A61P35/00;C07D403/06;C07D405/06;C07D409/06;C07D413/12;C07D413/14;C07D417/06;C07D417/12;C07D417/14

主分类号:C07D413/06

摘要:A compound represented by the formula (I) or a salt of the compound, and a PPAR-.delta. activator which contains the compound or salt as the active ingredient: (see formula I) (wherein A represents O or S; B1 represents N, etc.; B2 represents O, etc.; each of X1 and X2 represents O, S, a bond, etc.; Y represents C1-8 alkylene chain; Z represents O or S; R1 represents aryl, etc. which can have substituents; R2 represents C1-8 alkyl, etc.; R3 represents C1-8 alkyl, C2-8 alkenyl, etc.; each of R4 and R5 represents hydrogen, C1-8 alkyl, etc.; and R6 represents hydrogen, etc.; provided that each of Z and R3 is attached to the benzene ring, and X2 is not attached to the benzene ring).

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