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Composés de 6-benzyl-2, 3,4, 7-tétrahydro-indolo [2, 3-c] quinoline utiles en tant qu'inhibiteurs de pde5

申请公布号:MA31229(B1)

申请号:MA20090032183

申请日期:2009.08.31

申请公布日期:2010.03.01

申请人:
NYCOMED GMBH

发明人:WEINBRENNER, STEFFEN;DUNKERN, TORSTEN;MARX, DEGENHARD;SCHMIDT, BEATE;STENGEL, THOMAS;FLOCKERZI, DIETER;KAUTZ, ULRICH;HAUSER, DANIELA;DIEFENBACH, JÖRG;CHRISTIAANS, JOHANNES A. M.;MENGE, WIRO M.P.B.

分类号:C07D471/04;A61K31/437;A61P9/00;A61P15/00;A61P25/00;A61P29/00;(IPC1-7):C07D471/04

主分类号:C07D471/04

摘要:L'invention concerne des composés de formule (i) dans laquelle r1 à r8 et r11 sont tels que décrits dans la description, leurs sels, les n-oxydes de ces composés et leurs sels, et les stéréoisomères de ces composés, les sels, les n-oxydes de ces composés et les n-oxydes de leurs sels sont des inhibiteurs efficaces de la phosphodiestérase de type 5.

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