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DIAZA HETEROCYCLIC SULFONAMIDE DERIVATIVES AND THEIR USES

申请公布号:WO2007070506(A2)

申请号:WO2006US47353

申请日期:2006.12.13

申请公布日期:2007.06.21

申请人:
AMGEN INC.;POWERS, JAY, P.;SUN, DAQING;TU, HUA;YAN, XUELEI

发明人:POWERS, JAY, P.;SUN, DAQING;TU, HUA;YAN, XUELEI

分类号:C07D295/22;A61K31/496;A61P3/06;C07D401/04;C07D403/06

主分类号:C07D295/22

摘要:Diaza heterocyclic sulfonamide derivatives according to formula I have therapeutic utility, particularly in the treatment of diabetes, obesity and related conditions and disorders: I where R<SUP>7</SUP>, R<SUP>8</SUP>, R<SUP>9</SUP>, R<SUP>10</SUP>, R<SUP>11</SUP>, R<SUP>12</SUP>, R<SUP>13</SUP>, X, Y<SUP>1</SUP>, Y<SUP>2</SUP>, m, and n are set forth in the description.

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