Uudne protsess N-[(S)-1-karboksübutüül]-(S)-alaniini estrite sünteesimiseks ning nende rakendamine perindopriili sünteesis
申请公布号:EE200200553(A)
申请号:EE20020000553
申请日期:2001.03.30
申请公布日期:2004.04.15
发明人:JEAN-CLAUDE SOUVIE
分类号:C07C227/18;A61P9/00;C07B61/00;C07C22/00;C07C227/32;C07C229/16;C07C229/24;C07D209/34;(IPC1-7):C07C227/32
主分类号:C07C227/18
摘要:<p>Stereoselective process for the industrial synthesis of compounds of formula (I):wherein R represents linear or branched (C1-C6)alkyl.Application in the synthesis of perindopril and pharmaceutically acceptable salts thereof.</p>