用于抗菌的2-羟基-姆替林氨基甲酸酯衍生物
申请公布号:CN1427827A
申请号:CN01809198.9
申请日期:2001.03.29
申请公布日期:2003.07.02
发明人:杰拉尔德·布鲁克斯;埃里克·亨特;史蒂文·霍华德
分类号:C07D239/42;A61K31/44;A61K31/425;A61P31/04;C07D213/81;C07D277/56;C07D417/04;C07D487/04
主分类号:C07D239/42
代理人:黄益芬;巫肖南
地址:英国米德尔塞克斯
摘要:式(I)的2-(S)-羟基姆替林(mutilin)氨基甲酸酯衍生物,其中R<SUP>1</SUP>是5-或6-元的可被取代或不被取代的杂芳基;以及R<SUP>2</SUP>是乙烯基或乙基,该化合物可用于治疗细菌性感染。
主权项:1、式(I)化合物:<img file="A0180919800021.GIF" wi="1150" he="565" />其中:R<sup>1</sup>为可被取代或不被取代的5-或6-元杂芳基;和R<sup>2</sup>为乙烯基或乙基。
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