Novel pyrimidine derivative and novel pyridine derivative
申请公布号:AU8450401(A)
申请号:AU20010084504
申请日期:2001.09.10
申请公布日期:2002.03.26
发明人:SEIJI OHNO;KAYO OTANI;SEIJI NIWA;SATOSHI IWAYAMA;AKIRA TAKAHARA;HAJIME KOGANEI;YUKITSUGU ONO;SHINICHI FUJITA;TOMOKO TAKEDA;MASAKO HAGIHARA;AKIKO OKAJIMA
分类号:A61K31/455;A61K31/496;A61K31/505;A61K31/506;A61K31/5377;A61K31/55;A61K31/551;A61P1/04;A61P9/10;A61P11/06;A61P25/00;A61P25/04;A61P25/06;A61P25/16;A61P25/28;A61P25/30;A61P43/00;C07D213/80;C07D213/82;C07D239/28;C07D239/34;C07D239/38;C07D239/42;C07D401/04;C07D403/04;C07D409/04;C07D417/04
主分类号:A61K31/455
摘要:Achiral pyrimidine derivatives and pyridine derivatives of the following formulae or analogs thereof have selective N-type calcium channel antagonistic activity and showed analgesic action when they were taken orally. They are useful as therapeutic agents for pains and various diseases associated with the N-type calcium channels. <CHEM> <CHEM>