Tetrahydronapthalene derivatives and their therapeutic use
申请公布号:US6133240(A)
申请号:US19970924688
申请日期:1997.09.05
申请公布日期:2000.10.17
发明人:TAYLOR, RICHARD JOHN KENNETH;MURPHY, PAUL VINCENT;MONTANA, JOHN GARY;MANALLACK, DAVID THOMAS
分类号:A61K31/704;A61P1/00;A61P9/10;A61P11/02;A61P11/06;A61P17/00;A61P17/06;A61P19/02;A61P27/00;A61P29/00;A61P31/18;A61P43/00;C07H15/203;(IPC1-7):A61K31/70;C07H15/00
主分类号:A61K31/704
摘要:Compounds of the formula wherein R1 is a fucose or mannose residue, have therapeutic utility via inhibition of selectins, and thus of cell adhesion.