PROCESS FOR THE PREPARATION OF RIBONUCLEOTIDE REDUCTASE INHIBITORS.
申请公布号:MX9500363(A)
申请号:MX19950000363
申请日期:1995.01.06
申请公布日期:1998.04.30
发明人:RICHARD E. DONALDSON
分类号:A61K31/70;A61K31/7042;A61K31/7052;A61K31/7064;A61K31/7068;A61P31/12;A61P35/00;A61P43/00;C07D405/04;C07H19/06;(IPC1-7):C07D307/00
主分类号:A61K31/70
摘要:The present invention is directed toward a novel process of preparing 2'-exocyclic vinylfluoride derivatives of cytidine analogues for use as ribonucleotide reductase inhibitors.