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Substituted phthalazinones as neurotensin antagonists

申请公布号:US5668279(A)

申请号:US19950411655

申请日期:1995.04.06

申请公布日期:1997.09.16

申请人:
MERCK & CO., INC.

发明人:CHAKRAVARTY, PRASUN K.;NAYLOR, ELIZABETH M.;CHEN, ANNA

分类号:A61K31/50;A61K31/502;A61P1/00;A61P1/04;A61P1/12;A61P25/18;A61P25/24;A61P25/26;A61P25/28;C07D237/32;C07D401/04;C07D405/12;C07D409/12;(IPC1-7):C07D237/32;C07D409/04;C07D413/10

主分类号:A61K31/50

摘要:PCT No. PCT/US93/10386 Sec. 371 Date Apr. 6, 1995 Sec. 102(e) Date Apr. 6, 1995 PCT Filed Oct. 28, 1993 PCT Pub. No. WO94/10151 PCT Pub. Date May 11, 1994Novel substituted phthalazinones of the formula (I) <IMAGE> are useful as neurotensin antagonists.

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