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TRANSOCULAR PHARMACEUTICAL PREPARATION

申请公布号:CA2119233(A1)

申请号:CA19922119233

申请日期:1992.09.16

申请公布日期:1993.04.01

申请人:
FUJISAWA PHARMACEUTICAL CO

发明人:SHIMOJO FUMIO;SAWAI SEIJI;HORI SADAO;KOSEKI YOSHIYUKI;TERANO HIROSHI;OKUHARA MASAKUNI

分类号:A61K9/00;A61K31/335;(IPC1-7):A61K31/335;A61K9/06;A61K9/08

主分类号:A61K9/00

摘要:The ophthalmic pharmaceutical preparation of the present invention comprises oxaspirooctane derivatives (I) represented by the general formula: <IMG> (I) wherein R1 is carbamoyl; R2 is lower alkoxy; and R3 is represented by the following formula: <IMG> or salts thereof as an active ingredient and pharmaceutically acceptable carrier(s). 26

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